- Search results for Cay11731
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10 products were found matching "Cay11731"!
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Item number: Cay11731-10
Bosentan is an antagonist of the endothelin receptors type A (Ki = 6.5 nM) and type B (Ki = 340 nM).Formal Name: 4-(1,1-dimethylethyl)-N-[6-(2-hydroxyethoxy)-5-(2-methoxyphenoxy)[2,2'-bipyrimidin]-4-yl]-benzenesulfonamide. CAS Number: 147536-97-8. Synonyms: Ro 47-0203. Molecular Formula: C27H29N5O6S. Formula Weight:...
Keywords: | Ro 47-0203, 4-(1,1-dimethylethyl)-N-[6-(2-hydroxyethoxy)-5-(2-methoxyphenoxy)[2,2'-bipyrimidin]-4-yl]-benzenesulfonamide |
Application: | Endothelin receptor antagonist |
CAS | 147536-97-8 |
MW: | 551.6 D |
From 44.00€
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Item number: Cay11773-1
UR-144 (Cay-11502) is a potent synthetic cannabinoid (CB) which preferentially binds the peripheral CB2 receptor (Ki = 1.8 nM) over the central CB1 receptor (Ki = 150 nM). UR-144 N-pentanoic acid metabolite is an expected phase I metabolite of UR-144, based on the metabolism of similar cannabimimetics. This...
Keywords: | XLR11 N-pentanoic acid metabolite, 3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indole-1-pentanoic acid |
Application: | Analytical reference standard, Expected phase I UR-144 metabolite |
CAS | 1451369-33-7 |
MW: | 341.5 D |
From 158.00€
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Item number: Cay11173-1
Glucose transporter 1 (Glut1) is an inducible carrier of pentoses and hexoses, including glucose. STF-31 is an inhibitor of Glut1 (IC50 = ~1 µM) that blocks glucose uptake. It induces necrosis in cancer cells that lack the von Hippel-Lindau tumor suppressor gene, which overexpress Glut1. Although STF-31 binds Glut1,...
Keywords: | 4-[[[[4-(1,1-dimethylethyl)phenyl]sulfonyl]amino]methyl]-N-3-pyridinyl-benzamide |
Application: | GLUT1 inhibitor |
CAS | 724741-75-7 |
MW: | 423.5 D |
From 60.00€
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Item number: Cay11733-1
Atazanavir is an azapeptide inhibitor of HIV-1 protease (Ki = 2.66 nM). It has antiviral activity against a variety of HIV-1 strains in several cell types with EC50 values ranging from 2.62 to 5.28 nM. Atazanavir exhibits a minor synergistic effect when used in combination with the reverse transcriptase inhibitor...
Keywords: | BMS 232632, CGP 73547,... |
Application: | HIV-1 protease inhibitor |
CAS | 198904-31-3 |
MW: | 704.9 D |
From 49.00€
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Item number: Cay17333-1
Temoporfin is a synthetic chlorin with light-activated actions. When administered systemically, temoporfin accumulates in tumor cells. When stimulated with light (650-652 nm) in the presence of oxygen, reactive oxygen species are generated, leading to necrosis within the tumor. Different approaches to using...
Keywords: | m-THPC, Foscan, KW 2345, 3,3',3'',3'''-(7,8-dihydro-21H,23H-porphine-5,10,15,20-tetrayl)tetrakis-phenol |
Application: | Light-activated necrosis inducer |
CAS | 122341-38-2 |
MW: | 680.8 D |
From 43.00€
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Item number: Cay17733-1
Quinacrine analog 34 is an inhibitor of autophagy with a minimum effective concentration (MEC) of 0.5 µM in U2OS cells. It induces lysosomal deacidification and accumulation of LC3-II in the same cells when used at concentrations of 0.5 or 3 µM.Formal Name:...
Keywords: | 6-chloro-1,2,3,4-tetrahydro-N-[2-(4-methyl-1-piperazinyl)ethyl]-9-acridinamine |
Application: | Autophagy inhibitor |
CAS | 1411646-44-0 |
MW: | 358.9 D |
From 84.00€
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Item number: Cay17331-5
5,7-dichloro Tryptamine is a ring-substituted tryptamine derivative. Although the biological effects of this compound have not been reported, tryptamines substituted with fluorine at the 5-, 6-, or 7-position have been shown to have 5-HT2C receptor selectivity over both the 5-HT2A and 5-HT2B subtypes. This product...
Keywords: | 5,7-dichloro-1H-indole-3-ethanamine, monohydrochloride |
Application: | Analytical reference standard, Ring-substituted tryptamine derivative |
CAS | 94850-28-9 |
MW: | 265.6 D |
From 60.00€
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Item number: Cay11738-1
LY320135 is a selective cannabinoid (CB) receptor 1 antagonist (Kis = 224 and >10,000 nM for CB1 and CB2, respectively, in vitro). It is selective for CB1 over alpha1- and alpha2- adrenergic, D1 and D2 dopamine, benzodiazepine, histamine H1, GABA, serotonin (5-HT), and muscarinic receptors. It reverses the...
Keywords: | 4-[[6-methoxy-2-(4-methoxyphenyl)-3-benzofuranyl]carbonyl]-benzonitrile |
Application: | Cannabinoid receptor 1 (CB1) antagonist |
CAS | 176977-56-3 |
MW: | 383.4 D |
From 39.00€
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Item number: Cay11730-1
Coumestrol is a phytoestrogen that occurs naturally in soybeans, spinach, and clover. It competitively (vs. 17beta-estradiol, Cay-10006315) binds the estrogen receptors ERalpha (IC50 = 11 nM) and ERbeta (IC50 = 2 nM) and can induce ER-dependent gene expression in isolated cells. Coumestrol is also a weak antagonist...
Keywords: | NSC 22842, 3,9-dihydroxy-6H-benzofuro[3,2-c][1]benzopyran-6-one |
Application: | Pregnane X receptor antagonist |
CAS | 479-13-0 |
MW: | 268.2 D |
From 60.00€
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Item number: Cay11739-1
Makisterone A is an ecdysteroid that drives molting in insects. It binds the heterodimeric ecdysone receptor with nanomolar affinity.Formal Name: (2beta,3beta,5beta,22R,24R)-2,3,14,20,22,25-hexahydroxy-ergost-7-en-6-one. CAS Number: 20137-14-8. Molecular Formula: C28H46O7. Formula Weight: 494.7. Purity: >95%....
Keywords: | (2beta,3beta,5beta,22R,24R)-2,3,14,20,22,25-hexahydroxy-ergost-7-en-6-one |
Application: | Ecdysone receptor agonist |
CAS | 20137-14-8 |
MW: | 494.7 D |
From 49.00€
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