3 products were found matching "Cay11038"!

No results were found for the filter!
Bafilomycin A1
Bafilomycin A1

Item number: Cay11038-500

Bafilomycin A1 is a bacterial metabolite that has been found in Streptomyces and has diverse biological activities. It is an inhibitor of vacuolar H+-ATPases (V-ATPases, Ki = 0.5 nM in N. crassa vacuolar membranes) and is greater than 1,000-fold selective for V-ATPases over Na+/K+-, Ca2+-, and H+-ATPases....
Keywords: NSC 381866,...
Application: V-ATPase inhibitor
CAS 88899-55-2
MW: 622.8 D
From 125.00€ *
Review
TMS
TMS

Item number: Cay10038-1

CYP1B1 is mainly an extrahepatic enzyme which oxidatively metabolizes both endogenous (steroids, eicosanoids) and exogenous xenobiotics such aspolyaromatic hydrocarbons. TMS is a potent and selective inhibitor of CYP1B1, with an IC50 of 6 nM. It is 50-fold selective for the inhibition of CYP1B1 versus CYP1A1, making...
Keywords: 2,3',4,5'-Tetramethoxystilbene, 1-[(1E)-2-(3,5-dimethoxyphenyl)ethenyl]-2,4-dimethoxy-benzene
Application: CYP1B1 inhibitor
CAS 24144-92-1
MW: 300.4 D
From 22.00€ *
Review
Naringenin-7-O-beta-D-Glucuronide
Naringenin-7-O-beta-D-Glucuronide

Item number: Cay10388-5

Naringenin-7-O-beta-D-glucuronide is a metabolite of the flavonoid naringenin (Cay-14173). It is formed from naringenin primarily by the UDP-glucuronosyltransferase (UGT) isoforms UGT1A1, UGT1A3, UGT1A6, and UGT1A9.Formal Name: 3,4-dihydro-5-hydroxy-2-(4-hydroxyphenyl)-4-oxo-2H-1-benzopyran-7-yl,...
Keywords: (2S)-3,4-dihydro-5-hydroxy-2-(4-hydroxyphenyl)-4-oxo-2H-1-benzopyran-7-yl-beta-D-glucopyranosiduronic acid
Application: CYP1A2 inhibitor
CAS 1237479-07-0
MW: 448.4 D
From 172.00€ *
Review