5 products were found matching "Cay11787"!

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BRD4770
BRD4770

Item number: Cay11787-25

BRD4770 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, decreasing di- and trimethylation on lysine 9 of histone 3 (EC50 = 5 µM). Through its effects on EHMT2, BRD4770 induces senescence in the pancreatic cancer cell line PANC-1 without initiating apoptosis. It also blocks both...
Keywords: HMTase Inhibitor VI, 2-(benzoylamino)-1-(3-phenylpropyl)-1H-benzimidazole-5-carboxylic acid, methyl ester
Application: EHMT2 inhibitor
CAS 1374601-40-7
MW: 413.5 D
From 43.00€ *
Review
IAA-94
IAA-94

Item number: Cay17877-10

IAA-94 is an indanyloxyacetic acid (IAA) inhibitor of chloride channels that binds channels in bovine kidney cortex microsomes with a Ki value of 1 µM. At 10 µM, it also reversibly inhibits chloride intracellular channel proteins, which have both soluble and membrane-bound activities. IAA-94 is used to study the...
Keywords: R(+)-IAA 94, 2-[[(2R)-6,7-dichloro-2-cyclopentyl-2,3-dihydro-2-methyl-1-oxo-1H-inden-5-yl]oxy]-acetic acid
Application: Chloride channel inhibitor
CAS 54197-31-8
MW: 357.2 D
From 50.00€ *
Review
Bambuterol (hydrochloride)
Bambuterol (hydrochloride)

Item number: Cay17887-100

Bambuterol is a prodrug form of the beta-adrenergic receptor (beta-AR) agonist terbutaline (Cay-29337). It is also an inhibitor of butyrylcholinesterase (BChE, IC50 = 3.9 nM for the human enzyme), the enzyme that metabolizes bambuterol into terbutaline, and this inhibition increases the duration of action of...
Keywords: KWD 2183, N,N-dimethyl-carbamic...
Application: BCHE substrate, long-acting beta-adrenoceptor agonist agonist
CAS 81732-46-9
MW: 403.9 D
From 43.00€ *
Review
MAM2201 N-(4-hydroxypentyl) metabolite
MAM2201 N-(4-hydroxypentyl) metabolite

Item number: Cay11778-1

MAM2201 (Cay-9001219) is a synthetic cannabinoid (CB) that is closely related, structurally, to AM2201 (Cay-10707), a compound which displays high affinities for both CB receptors. MAM2201 N-(4-hydroxypentyl) metabolite is a potential phase 1 metabolite of MAM2201, based on the known metabolism of similar compounds....
Keywords: [1-(5-fluoro-4-hydroxypentyl)-1H-indol-3-yl](4-methyl-1-naphthalenyl)-methanone
Application: Analytical reference standard, potential phase I MAM2201 metabolite
CAS 1537889-05-6
MW: 389.5 D
From 109.00€ *
Review
AB-005 azepane isomer
AB-005 azepane isomer

Item number: Cay11877-10

AB-005 (Cay-11766) is a synthetic cannabinoid (CB) built on a 1-[(1-methylpiperidin-2-yl)methyl]-indole base that is characteristic of a series of potent CBs, including AM1220 (Cay-9001055), AM1241 (Cay-10010118), and AM1248 (Cay-11282). AB-005 azepane isomer is a variant of AB-005 in which the methylpiperidine...
Keywords: [1-(hexahydro-1-methyl-1H-azepin-3-yl)-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)-methanone
Application: Analytical reference standard, Synthetic cannabinoid variant
CAS 1445751-74-5
MW: 352.5 D
From 109.00€ *
Review