8 products were found matching "Cay16516-500"!
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BRD32048
Item number: Cay16516-5
ETS variant 1 (ETV1) is a transcription factor oncogene implicated in several cancers where it has been altered by chromosomal translocation, gene amplification, or lineage dysregulation. The ETV1 transcription factor is phosphorylated downstream of MAPK signaling and is acetylated at lysines 33 and 116 by the...
| Keywords: | N2-(4-methoxyphenyl)-6-(1-piperidinylmethyl)-1,3,5-triazine-2,4-diamine |
| Application: | ETV1 inhibitor |
| CAS | 433694-46-3 |
| MW: | 314.4 D |
From 38.00€
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11-deoxy Prostaglandin F2beta
Item number: Cay16510-5
11-deoxy Prostaglandin F2beta (11-deoxy PGF2beta) is an analog of PGF2beta (Cay-16410).Formal Name: 9beta,15S-dihydroxy-prosta-5Z,13E-dien-1-oic acid. CAS Number: 37786-07-5. Synonyms: 11-deoxy PGF2beta. Molecular Formula: C20H34O4. Formula Weight: 338.5. Purity: >98%. Formulation: (Request formulation change), A...
| Keywords: | 11-deoxy PGF2beta, 9beta,15S-dihydroxy-prosta-5Z,13E-dien-1-oic acid |
| Application: | Bioactive lipid assays |
| CAS | 37786-07-5 |
| MW: | 338.5 D |
From 86.00€
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5-Azidopentanoic Acid
Item number: Cay16517-500
5-Azidopentanoic acid is a building block for use in click chemistry reactions that enables selective conjugation of peptides with various molecules and can be used for the cyclization of peptides. The azido moiety reacts with acetylenes in the presence of copper yielding triazoles that can function as versatile...
| Keywords: | 5-Azidovaleric acid, Click Tag(TM) 5-Azidopentanoic Acid, 5-azido-pentanoic acid |
| Application: | Building block, Click Chemistry |
| CAS | 79583-98-5 |
| MW: | 143.1 D |
From 146.00€
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4-fluoro-alpha-Pyrrolidinopentiophenone (hydrochloride)
Item number: Cay15166-50
alpha-Pyrrolidinopentiophenone (alpha-PVP, Cay-9001083) is an analog of pyrovalerone (Cay-10817), a known monoamine transport inhibitor that prevents the reuptake of dopamine and norepinephrine. 4-fluoro-alpha-PVP is an isomer of alpha-PVP characterized by the addition of a fluorine group at the 4 position of the...
| Keywords: | 4-fluoro-alpha-PVP, 4-fluoro-2-(1-pyrrolidinyl)-Valerophenone, 4-fluoro-alpha-Pyrrolinovalerophenone,... |
| Application: | Analytical reference standard, Pyrovalerone analog |
| CAS | 850352-31-7 |
| MW: | 285.8 D |
From 291.00€
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Eplerenone
Item number: Cay15616-50
Eplerenone is a mineralocorticoid receptor antagonist. It is selective for the mineralocorticoid receptor over glucocorticoid, androgen, progesterone, and estrogen receptors in radioligand binding assays (IC50s = 138, 6,920, 523, >10,000, and 5,702 nM, respectively). Eplerenone inhibits aldosterone-induced...
| Keywords: | (+)-Eplerenone, CGP 30083, Epoxymexrenone, SC-6110, SC-66110,... |
| Application: | Mineralocorticoid receptor antagonist |
| CAS | 107724-20-9 |
| MW: | 414.5 D |
From 84.00€
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Estradiol 17-(beta-D-Glucuronide) (sodium salt hydrate)
Item number: Cay16156-50
Estradiol 17-(beta-D-glucuronide) (E217G) is an estrogen metabolite formed in the liver and subsequently excreted in bile. It acts as a substrate of the multidrug resistance protein 2 (MRP2, Km = 75 µM), and through MRP2-mediated transport, functions as a cholestatic agent, decreasing bile flow. In addition to...
| Keywords: | 17beta-Estradiol 17-(beta-D-Glucuronide), 17beta-Oestradiol 17-(beta-D-Glucuronide), E217G, beta-Estradiol... |
| Application: | ABCC2 substrate |
| MW: | 470.5 D |
From 98.00€
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Ketoconazole-d3
Item number: Cay10010656-500
Ketoconazole-d3 is intended for use as an internal standard for the quantification of ketoconazole (Cay-15212) by GC- or LC-MS. Ketoconazole is a broad-spectrum triazole antifungal agent that has activity against C. albicans, C. krusei, C. tropicalis, C. glabrata, C. parapsilosis, C. neoformans, and A. fumigatus...
| Keywords: | 1-(4-(4-(((2R,4S)-2-((1H-imidazol-1-yl)methyl)-2-(2,4-dichlorophenyl)-1,3-dioxolan-4-yl)methoxy)phenyl)piperazin-1-yl)etha... |
| Application: | GC-MS, LC-MS, Quantification, Internal standard |
| CAS | 1217766-70-5 |
| MW: | 534.5 D |
From 43.00€
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PF-04418948
Item number: Cay15016-50
Prostaglandin E2 (PGE2) evokes distinct responses through four different 'E prostanoid' (EP) receptors. EP2 is a G protein-coupled receptor which signals preferentially through Gs proteins. PF-04418948 is an orally active, potent, and selective EP2 receptor antagonist (IC50 = 16 nM). It is over a thousand-fold less...
| Keywords: | 1-(4-fluorobenzoyl)-3-[[(6-methoxy-2-naphthalenyl)oxy]methyl]-3-azetidinecarboxylic acid |
| Application: | EP2 receptor antagonist |
| CAS | 1078166-57-0 |
| MW: | 409.4 D |
From 131.00€
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