6 products were found matching "Cay13705"!
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Halofuginone (hydrochloride)
Item number: Cay13370-5
Halofuginone is a halogenated derivative of febrifugine, a natural quinazolinone-containing compound found in the Chinese herb D. febrifuga. It has antimalarial and anticoccidial actions. In mammals, halofuginone at 10 ng/ml down-regulates Smad3, blocking TGF-beta signaling and preventing both the differentiation of...
| Keywords: | 7-bromo-6-chloro-3-[3-[(2R,3S)-3-hydroxy-2-piperidinyl]-2-oxopropyl]-4(3H)-quinazolinone, monohydrochloride |
| Application: | Antiprotozoal, glutamyl-prolyl-tRNA synthetase (EPRS) inhibitor, Smad3 down-regulator |
| CAS | 1217623-74-9 |
| MW: | 451.1 D |
From 163.00€
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2,3-MDMA (hydrochloride)
Item number: Cay13970-5
2,3-MDMA is an aromatic positional isomer of 3,4-MDMA (ecstasy, Cay-13971), a euphoric entactogen that is illegal in most countries and is regulated (Schedule I) in the United States. While 2,3-MDMA exhibits a similar potency to 3,4-MDMA for inhibition of the noradrenalin transporter (IC50s = 6.2 and 6.6 µM,...
| Keywords: | 2,3-Methylenedioxymethylamphetamine, N,alpha-dimethyl-1,3-benzodioxole-4-ethanamine, monohydrochloride |
| Application: | Analytical reference standard, Aromatic positional 3,4-MDMA isomer |
| CAS | 168968-01-2 |
| MW: | 229.7 D |
From 232.00€
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Butaprost
Item number: Cay13740-5
Butaprost, a structural analog of PGE2, is a selective agonist for the EP2 receptor subtype. EP2 receptors are expressed on human neutrophils and on respiratory, vascular, and uterine smooth muscle. Butaprost binds with about 1/10 the affinity of PGE2 to the recombinant murine EP2 receptor, and does not bind...
| Keywords: | 15-deoxy-16S-hydroxy-17-cyclobutyl PGE1 methyl ester, TR 4979,... |
| Application: | EP2 receptor agonist |
| CAS | 69685-22-9 |
| MW: | 408.6 D |
From 115.00€
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Pyroxamide
Item number: Cay13870-5
Pyroxamide is an inhibitor of histone deacetylases (HDACs), including HDAC1 (IC50 = 0.1-0.2 µM). It induces growth suppression and cell death of certain types of cancer cells in culture.Formal Name: N1-hydroxy-N8-3-pyridinyl-octanediamide. CAS Number: 382180-17-8. Molecular Formula: C13H19N3O3. Formula Weight:...
| Keywords: | N1-hydroxy-N8-3-pyridinyl-octanediamide |
| Application: | Histone deacetylases Inhibitor |
| CAS | 382180-17-8 |
| MW: | 265.3 D |
From 82.00€
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15(R)-Prostaglandin E1
Item number: Cay13710-5
15(R)-PGE1 is the "unnatural" C-15 stereoisomer of PGE1. It is essentially inactive biologically when compared to PGE1. It is a non-competitive inhibitor of 15-hydroxy PGDH with an IC50 of 189 µM.Formal Name: 9-oxo-11alpha,15R-dihydroxy-prost-13E-en-1-oic acid. CAS Number: 20897-91-0. Synonyms: 15(R)-PGE1, 15-epi...
| Keywords: | 15(R)-PGE1, 15-epi PGE1, 9-oxo-11alpha,15R-dihydroxy-prost-13E-en-1-oic acid |
| Application: | PGDH inhibitor |
| CAS | 20897-91-0 |
| MW: | 354.5 D |
From 97.00€
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GPP 78
Item number: Cay13670-5
Nicotinamide phosphoribosyltransferase (Nampt) converts nicotinamide into nicotinamide mononucleotide (NMN), which is subsequently converted to NAD+ by NMN adenyltransferase. Cancer cells commonly have an unusually high rate of NAD+ turnover, suggesting that inhibition of Nampt might selectively target cancer cells....
| Keywords: | CAY10618, NMPRTase Inhibitor, N-[1,1'-biphenyl]-2-yl-4-(3-pyridinyl)-1H-1,2,3-triazole-1-octanamide |
| Application: | NAMPT inhibitor |
| CAS | 1202580-59-3 |
| MW: | 439.6 D |
From 27.00€
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