6 products were found matching "Cay14715"!

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AMG 9810
AMG 9810

Item number: Cay14715-10

AMG 9810 is a competitive antagonist of capsaicin activation of the vanilloid receptor 1 (TRPV1) (IC50s = 24.5 and 85.6 nM for human and rat, respectively). Additionally, it has been shown to compete with other modes of TRPV1 activation, including protons (IC50s = 92.7 and 294 nM for human and rat, respectively),...
Keywords: (2E)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[4-(1,1-dimethylethyl)phenyl]-2-propenamide
Application: TRPV1 antagonist
CAS 545395-94-6
MW: 337.4 D
From 77.00€ *
Review
2C-TFM (hydrochloride)
2C-TFM (hydrochloride)

Item number: Cay14471-5

A series of 2,5-dimethoxyphenethylamines, collectively referred to as 2Cs, have psychoactive effects. The most effective 2C compounds are substituted at the 4 position of the aromatic ring, many are scheduled as illegal substances. 2C-TFM is a 2C compound with a para-trifluoromethyl substitution. It is a potent...
Keywords: 2C-CF3, 2,5-dimethoxy-4-(trifluoromethyl)-benzeneethanamine, monohydrochloride
Application: Analytical reference standard, Potent 5-HT2A / 5-HT2C agonist
CAS 159277-13-1
MW: 285.7 D
From 266.00€ *
Review
15(R)-Prostaglandin E2
15(R)-Prostaglandin E2

Item number: Cay14710-5

15(R)-Prostaglandin E2 (15(R)-PGE2) is the C-15 epimer of the naturally occurring 15(S)-PGE2. 15(R)-PGE2 is much less potent than the natural stereoisomer in most biological assays. In hamsters, a dose of 0.20 mg of PGE2 (Cay-14010) inhibits fertility by 100%, whereas a dose of 1.0 mg of 15(R)-PGE2 inhibits...
Keywords: 15(R)-PGE2, 15-epi PGE2, 9-oxo-11alpha,15R-dihydroxy-prosta-5Z,13E-dien-1-oic acid
Application: Bioactive lipid assays
CAS 38873-82-4
MW: 352.5 D
From 86.00€ *
Review
Aprotinin
Aprotinin

Item number: Cay14716-25

Aprotinin is a reversible inhibitor of serine proteases such as trypsin (Ki = 0.06 pM), chymotrypsin (Ki = 9.5 nM), and kallikrein (Ki = 0.8 nM). It is a much weaker inhibitor of thrombin (Ki = 0.1-0.8 mM) and trypsinogen (Ki = 2 µM). Aprotinin also competitively inhibits nNOS and iNOS with Ki values of 50 and 78...
Keywords: Bovine Pancreatic Trypsin Inhibitor, BPTI
Application: Serine protease inhibitor, protein purification
CAS 9087-70-1
MW: 6511.4 D
From 39.00€ *
Review
Dimethyl fumarate
Dimethyl fumarate

Item number: Cay14714-25

Dimethyl fumarate is a lipophilic electrophile that has profound effects on oxidative and immunological pathways. It rapidly interacts in a Michael addition reaction with glutathione or is metabolized to monomethyl fumarate. Dimethyl fumarate at low micromolar levels activates the nuclear factor erythroid 2-related...
Keywords: trans-Butenedioic Acid dimethyl ester, NSC 167432, NSC 25942, 2E-butenedioic acid, 1,4-dimethyl ester
Application: Nrf2 activator
CAS 624-49-7
MW: 144.1 D
From 31.00€ *
Review
Sophorose
Sophorose

Item number: Cay14717-25

Sophorose is a disaccharide component of the microbial glycolipids produced by yeast termed sophorolipids. Due to their hydrophobic nature, sophorolipids are often employed as biosurfactants. Sophorolipids also demonstrate antibacterial, antifungal, spermicidal, virucidal, and anti-cancer activities. Sophorose has...
Keywords: 2-O-beta-D-glucopyranosyl-D-glucose
Application: Disaccharide, Cellulase gene expression inducer
CAS 20429-79-2
MW: 342.3 D
From 270.00€ *
Review