9 products were found matching "Cay37720"!

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15(S)-HEDE
15(S)-HEDE

Item number: Cay37720-50

15(S)-HEDE is produced from 11Z,14Z-eicosadienoic acid by 15-LO. 15(S)-HEDE is an inhibitor of RBL-1 cell 5-LO with an IC50 value of 26 µM.Formal Name: 15S-hydroxy-11Z,13E-eicosadienoic acid. CAS Number: 92693-04-4. Molecular Formula: C20H36O3. Formula Weight: 324.5. Purity: >98%. Formulation: (Request formulation...
Keywords: 15S-hydroxy-11Z,13E-eicosadienoic acid
Application: 5-LO inhibitor
CAS 92693-04-4
MW: 324.5 D
From 158.00€ *
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Dipyanone (hydrochloride)
Dipyanone (hydrochloride)

Item number: Cay33720-1

Dipyanone (hydrochloride) (Cay-33720) is an analytical reference standard that is structurally similar to known opioids. This product is intended for research and forensic applications.Formal Name: 4,4-diphenyl-6-(1-pyrrolidinyl)-3-heptanone, monohydrochloride. CAS Number: 102762-20-9. Molecular Formula: C23H29NO ....
Keywords: N-pyrrolidino Methadone, 4,4-diphenyl-6-(1-pyrrolidinyl)-3-heptanone, monohydrochloride
Application: Analytical reference standard, Structurally similar to known opioids
CAS 102762-20-9
MW: 372 D
310.00€ *
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Sulfadoxin-d4
Sulfadoxin-d4

Item number: Cay37200-5

Sulfadoxin-d4 is intended for use as an internal standard for the quantification of sulfadoxin (Cay-21488) by GC- or LC-MS. Sulfadoxin is a sulfonamide antibiotic that inhibits dihydropteroate synthetase (DHPS), an enzyme involved in folic acid (Cay-20515) synthesis. Sulfadoxin competes with 4-aminobenzoate (PABA),...
Keywords: Ro 4-4393-d4, 4-amino-N-(5,6-dimethoxy-4-pyrimidinyl)-benzenesulfonamide-d4
Application: GC-MS, LC-MS, Internal standard, Quantification, Folic acid biosynthesis inhibitor
CAS 1330266-05-1
MW: 314.4 D
From 265.00€ *
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MCP110
MCP110

Item number: Cay37725-10

MCP110 is an inhibitor of the protein-protein interaction between Ras and Raf-1. It inhibits the interaction between H-Ras and Raf-1 in a yeast two-hybrid assay when used at a concentration of 30 µM. MCP110 (20 µM) inhibits Ras-induced activation of Raf-1 and MEK1 activity in HT-1080 fibrosarcoma cells. In vivo,...
Keywords: N-[[3-methoxy-4-(phenylmethoxy)phenyl]methyl]-N-[2-(2-pyridinyl)ethyl]-benzenepentanamide
Application: Ras-Raf-1 protein-protein interaction inhibitor
CAS 521310-51-0
MW: 508.7 D
From 47.00€ *
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Senaparib
Senaparib

Item number: Cay37722-10

Senaparib is an inhibitor of poly(ADP-ribose) polymerase 1 (PARP1) and PARP2.Formal Name: 5-fluoro-1-[[4-fluoro-3-[[4-(2-pyrimidinyl)-1-piperazinyl]carbonyl]phenyl]methyl]-2,4(1H,3H)-quinazolinedione. CAS Number: 1401682-78-7. Synonyms: IMP-4297. Molecular Formula: C24H20F2N6O3. Formula Weight: 478.5. Purity: >98%....
Keywords: IMP-4297, 5-fluoro-1-[[4-fluoro-3-[[4-(2-pyrimidinyl)-1-piperazinyl]carbonyl]phenyl]methyl]-2,4(1H,3H)-quinazolinedione
Application: PARP1 / PARP2 inhibitor
CAS 1401682-78-7
MW: 478.5 D
From 82.00€ *
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Tolebrutinib
Tolebrutinib

Item number: Cay37723-10

Tolebrutinib is an irreversible inhibitor of Bruton's tyrosine kinase (BTK, IC50 = 1 nM). It decreases the number of CD69+ B cells in isolated mouse whole blood (IC50 = 200 nM).Formal Name: 4-amino-1,3-dihydro-1-[(3R)-1-(1-oxo-2-propen-1-yl)-3-piperidinyl]-3-(4-phenoxyphenyl)-2H-imidazo[4,5-c]pyridin-2-one. CAS...
Keywords: 4-amino-1,3-dihydro-1-[(3R)-1-(1-oxo-2-propen-1-yl)-3-piperidinyl]-3-(4-phenoxyphenyl)-2H-imidazo[4,5-c]pyridin-2-one
Application: Irreversible BTK inhibitor
CAS 1971920-73-6
MW: 455.5 D
From 90.00€ *
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PfDHODH-IN-1
PfDHODH-IN-1

Item number: Cay37728-10

PfDHODH-IN-1 is an inhibitor of dihydroorotate dehydrogenase (DHODH, IC50s = 190, 47, and 21 nM for the human, mouse, and rat enzymes, respectively) and a derivative of the DHODH inhibitor A-771726 (Cay-14404). It inhibits delayed-type hypersensitivity reactions in mice and rats when administered at doses of 30 and...
Keywords: CCHTFP, PfDHODH Inhibitor 1, 2-cyano-3-cyclopropyl-3-hydroxy-N-[4-(trifluoromethyl)phenyl]-2-propenamide
Application: DHODH inhibitor
CAS 183945-55-3
MW: 296.2 D
From 35.00€ *
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ORG 41841
ORG 41841

Item number: Cay37724-10

ORG 41841 is a dual luteinizing hormone (LH) and thyroid-stimulating hormone (TSH) receptor agonist. It induces cAMP production in HEK293 cells expressing human LH or TSH receptors (EC50s = 0.3 and 6.5 µM, respectively).Formal Name:...
Keywords: 5-amino-N-(1,1-dimethylethyl)-4-(3-methoxyphenyl)-2-(methylthio)-thieno[2,3-d]pyrimidine-6-carboxamide
Application: Dual LH / TSH receptor agonist
CAS 301847-37-0
MW: 402.5 D
From 66.00€ *
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ERX-41
ERX-41

Item number: Cay37726-10

ERX-41 is an inducer of endoplasmic reticulum (ER) stress. It increases the thermal stability of lysosomal acid lipase when used at a concentration of 10 µM in the cellular thermal shift assay (CETSA) but does not inhibit lysosomal acid lipase enzymatic activity at 30 µM. ERX-41 (1 µM) increases ER tubule width,...
Keywords: 4-[[3-(2-hydroxyethoxy)-4-nitrobenzoyl]amino]-N-[4-[[(trans-4-methylcyclohexyl)amino]carbonyl]-2-(2-methylpropoxy)phenyl]-...
Application: ER stress inducer
CAS 2440087-54-5
MW: 704.8 D
From 117.00€ *
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