14 products were found matching "Cay34510-0.1"!

7-Fluoro-2,1,3-benzoxadiazole-4-sulfonate (SBD-F) is a thiol-reactive fluorogenic probe. It has been used to quantify the levels of homocysteine, cysteine, and cysteamine in human plasma. SBD-F displays excitation/emission maxima of 380/515 nm, respectively.Formal Name: 7-fluoro-2,1,3-benzoxadiazole-4-sulfonic acid,...

H-Arg-Gly-Asp-Cys-OH is a tetrapeptide that contains the arginine-glycine-aspartate (RGD) motif, a sequence that acts as a recognition site for various adhesion proteins. It inhibits the binding of fibrinogen to endothelial cells and ADP-stimulated platelets with IC50 values of 320 and 35 µM, respectively....

Benzetimide is a muscarinic acetylcholine receptor (mAChR) antagonist. It induces mydriasis and inhibits pilocarpine-induced salivation and lacrimation in rats (ED50s = 0.06 and 0.04 mg/kg, respectively).Formal Name: 3-phenyl-1'-(phenylmethyl)-[3,4'-bipiperidine]-2,6-dione, monohydrochloride. CAS Number: 5633-14-7....

Pendimethalin is a dinitroaniline herbicide. It controls johnsongrass and increases seed cotton yield when used at concentrations ranging from 0.56 to 1.12 kg/ha. Pendimethalin (25-500 µM) induces the production of reactive oxygen species (ROS) and genotoxicity in isolated human peripheral lymphocytes. In vivo,...

Picosulfate is a stimulant laxative and prodrug form of desacetyl bisacodyl (DAB, Cay-20928). Unlike bisacodyl (Cay-28826), picosulfate is hydrolyzed to DAB by colonic microbiota. Picosulfate (5 mg/kg) increases excreted fecal weight in a rat model of loperamide-induced constipation. Formulations containing...

Kanamycin B is an aminoglycoside antibiotic. It is active against S. aureus, E. coli, P. aeruginosa, and P. rettgeri (MICs = 0.78-25 µg/ml). Kanamycin B binds to the ribosomal decoding A site to interfere with bacterial protein synthesis.Formal Name:...

Naptalam is an auxin inhibitor and herbicide. It reduces coleoptile accumulation of the polar auxin indole-3-acetic acid (Cay-16954) in maize when used at a concentration of 50 µM. Naptalam inhibits various auxin-dependent processes, such as embryo development, lateral root development, leaf vein patterning, apical...

Glycine-d5 is intended for use as an internal standard for the quantification of glycine by GC- or LC-MS. Glycine is a conditionally essential amino acid and the major inhibitory neurotransmitter in the spinal cord and brainstem. It is synthesized from threonine, choline, hydroxyproline, and serine via interorgan...

(±)5-HETE lactone is a cyclic ester formed by acid-catalyzed nucleophilic addition of the C-5 hydroxyl to the C-1 carboxyl of (±)5-HETE. (±)5-HETE lactone is an inhibitor of 5-lipoxygenase from rat basophilic leukemia cells with an IC50 of 27 µM. The lactone is several times more potent than the linear...

Faropenem is a broad-spectrum penem antibiotic. It is active against a panel of 12 Gram-positive (MIC50s = 0.008-1 mg/L) and 15 Gram-negative (MIC50s = 0.06-16 mg/L) bacteria. Faropenem (20 mg/kg) reduces the number of lung colony forming units (CFUs) in a mouse model of H. influenzae-induced respiratory tract...

Dexmedetomidine is an agonist of alpha2-adrenergic receptors (alpha2-ARs). It selectively binds to alpha2-ARs over alpha1-ARs (Kis = 0.015 and 5 nM, respectively). In vivo, dexmedetomidine (50 µg/kg) prevents increases in cardiac troponin I (CTnI), a marker of myocardial injury, as well as reduces myocardial...

2-Aminotetralin is a neuromodulatory agent. It inhibits serotonin (5-HT) and norepinephrine reuptake in rat brain when administered at a dose of 39.4 mg/kg. 2-Aminotetralin induces hypothermia in rats when administered by intracisternal or intraperitoneal injection, but implantation of 2-aminotetralin crystals in...