- Search results for Cay10006794
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10 products were found matching "Cay10006794"!
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Item number: Cay10006974-5
AM630 binds selectively to cannabinoid 2 (CB2) over CB1 receptors with Ki values of 31.2 and 5,152 nM, respectively. AM630 acts as an inverse agonist at CB2 receptors, attenuating the antinociceptive effects of a number of cannabinoids, and as a weak partial agonist at CB1 receptors. It decreases proliferation and...
Keywords: | 6-Iodopravodoline, [6-iodo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](4-methoxyphenyl)-methanone |
Application: | CB2 receptor antagonist |
CAS | 164178-33-0 |
MW: | 504.4 D |
From 77.00€
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Lipid-based Drug Delivery Tools
Item number: Cay10007946-1
C16 Sphingomyelin is a naturally occurring sphingolipid. Levels of C16 sphingomyelin are elevated in the prefrontal cortex and cerebellum in a rat model of diabetes induced by streptozotocin (STZ, Cay-13104), as well as in the liver in mouse models of Niemann-Pick type C1 disease. Plasma levels of C16 sphingomyelin...
Keywords: | N-Palmitoyl-D-erythro-Sphingosylphosphorylcholine, Palmitoyl Sphingomyelin, SM(d18:1/16:0), Sphingomyelin (d18:1/16:0),... |
Application: | Bioactive Lipid Assays |
CAS | 6254-89-3 |
MW: | 703 D |
From 94.00€
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Item number: Cay10006798-5
The transcription factor peroxisome proliferator-activated receptor delta (PPARdelta) is a member of the superfamily of nuclear hormone receptors and is implicated both in lipid metabolism and in the regulation of genes with potential roles in neurotoxicity. GW 0742 is a selective PPARdelta agonist (EC50 = 1.1 nM)...
Keywords: | GW 610742, 2-[4-[[[2-[3-fluoro-4-(trifluoromethyl)phenyl]-4-methyl-5-thiazolyl]methyl]thio]-2-methylphenoxy]-acetic acid |
Application: | PPARdelta agonist |
CAS | 317318-84-6 |
MW: | 471.5 D |
From 109.00€
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Item number: Cay10006797-250
Xestospongins and araguspongins are marine natural products first isolated from Pacific basin sponges, and noted to have vasodilatory properties. Inositol phosphates (IP) are important signal transduction messengers acting via IP3 receptors to promote the mobilization of Ca2+ from intracellular stores. Araguspongin...
Keywords: | [1R-(1R*,4aR*,11S*,12aR*,13R*,16aR*,23S*,24aR*)]-eicosahydro-5H,17H-1,23:11,13-diethano-2H,14H-[1,11]dioxacycloeicosino[2,... |
Application: | IP3 receptor antagonist |
CAS | 123000-02-2 |
MW: | 446.7 D |
From 533.00€
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COVID-19 Research
Item number: Cay10007964-10
E-64c is an active metabolite of the protease inhibitor E-64d (Cay-13533). E-64c inhibits the cysteine proteases cathepsin B, cathepsin H, and papain but not the serine proteases trypsin, chymotrypsin, or elastase. It reduces the autocatalytic activity of the foot-and-mouth-disease virus (FMDV) leader protease when...
Keywords: | Loxistatin Acid, NSC 694279,... |
Application: | Cysteine protease inhibitor |
CAS | 76684-89-4 |
MW: | 314.4 D |
From 84.00€
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Item number: Cay10794-500
Agonists of the vitamin D receptor are used to suppress parathyroid hormone (PTH) synthesis and secretion in the treatment of hyperparathyroidism associated with renal failure. 22-Oxacalcitriol is an analog of calcitriol that, like calcitriol, is a receptor-active form of vitamin D3 which effectively blocks PTH...
Keywords: | Maxacalcitrol,... |
Application: | VDR ligand |
CAS | 103909-75-7 |
MW: | 418.6 D |
From 86.00€
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Item number: Cay10006790-1
ChREBP (carbohydrate response element-binding protein) is a transcription factor playing a critical role in the nutrient and hormonal regulation of genes encoding enzymes of glucose metabolism and lipogenesis pathways. It contains several domains including a nuclear localization signal (NSL) near the N-terminus,...
Keywords: | Carbohydrate Response Element-binding Protein, WBSCR14 |
Application: | Blocking |
177.00€
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Item number: Cay10006594-10
Losartan is an antagonist of angiotensin II type 1b (AT1b) receptor (IC50 = 2.2 nM in COS-7 cells expressing the rat receptor). It reduces U-46619-induced aggregation of platelets in isolated human platelet-rich plasma when used at a concentration of 5 µM. It decreases 1-lipoxygenase (1-LO) levels in the endothelial...
Keywords: | DuP-753, MK 954, 2-butyl-4-chloro-1-[[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4-yl]methyl]-1H-imidazole-5-methanol,... |
Application: | AT1 receptor antagonist |
CAS | 124750-99-8 |
MW: | 461 D |
From 23.00€
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Item number: Cay10006734-5
Nuclear factor-kappaB (NF-kappaB) is an ubiquitous transcription factor that functions to enhance the transcription of pro-inflammatory cytokines like TNF-alpha, IL-1beta, IL-6, and IL-8. QNZ is an inhibitor of NF-kappaB activation with an IC50 of 11 nM in human Jurkat cells. It also inhibits TNF-alpha production...
Keywords: | CAY10470, N4-[2-(4-phenoxyphenyl)ethyl]-4,6-quinazolinediamine |
Application: | NF-kappaB activation inhibitor |
CAS | 545380-34-5 |
MW: | 356.4 D |
From 27.00€
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Item number: Cay10006394-1
Formulation: HDAC developer.
Application: | Kit component |
28.00€
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