9 products were found matching "Cay10353"!

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SHS4121705
SHS4121705

Item number: Cay31053-5

SHS4121705 is an orally bioavailable mitochondrial uncoupler. It increases oxygen consumption rate in L6 rat myoblast cells with an EC50 value of 4.3 µM. SHS4121705 (25 mg/kg per day in the diet) reduces hepatic steatosis, liver triglyceride levels, and plasma alanine aminotransferase (ALT) levels in Stelic animal...
Keywords: 6-[[4-(trifluoromethoxy)phenyl]amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5(3H)-one
Application: Mitochondrial uncoupler
CAS 2379550-82-8
MW: 313.2 D
From 158.00€ *
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Prostaglandin F2alpha dimethyl amine
Prostaglandin F2alpha dimethyl amine

Item number: Cay16033-5

Prostaglandin F2alpha dimethyl amine (PGF2alpha dimethyl amine) is a derivative of PGF2alpha which was designed as a PG antagonist for in vitro and in vivo studies. PGF2alpha dimethyl amine is a weak FP receptor antagonist. In gerbil colon, PGF2alpha dimethyl amine at a dose of 3.2 µg/ml inhibits the contractile...
Keywords: Dinoprost dimethyl amine, PGF2alpha dimethyl amine, N,N,-dimethyl-9alpha,11alpha,15S-trihydroxy-prosta-5Z,13E-dien-1-amine
Application: FP receptor antagonist
CAS 67508-09-2
MW: 367.6 D
From 73.00€ *
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PRMT4/CARM1 Inhibitor
PRMT4/CARM1 Inhibitor

Item number: Cay11033-5

PRMT4/CARM1 Inhibitor selectively blocks the activity of PRMT4/CARM1 with an IC50 value of 7.1 µM. It displays very low affinity towards PRMT1 and SET7 with IC50 values of 63 and 943 µM, respectively. In human prostate cancer LNCaP cells, this compound reduced the prostate-specific antigen promoter activity at 8-10...
Keywords: Protein Arginine Methyltransferase 4/Coactivator-Associated Arginine Methyltransferase 1 Inhibitor,...
CAS 1020399-49-8
MW: 555.3 D
From 109.00€ *
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2-Fluorophenyl Cyclopentyl Ketone
2-Fluorophenyl Cyclopentyl Ketone

Item number: Cay31035-5

2-Fluorophenyl cyclopentyl ketone (Cay-31035) is an analytical reference standard categorized as a precursor in the synthesis of fluoroketamine. This product is intended for research and forensic applications.Formal Name: cyclopentyl(2-fluorophenyl)-methanone. CAS Number: 111982-45-7. Molecular Formula: C12H13FO....
Keywords: Cyclopentyl 2-Fluorophenyl Ketone, cyclopentyl(2-fluorophenyl)-methanone
Application: Analytical reference standard, fluoroketamine synthesis precursor
CAS 111982-45-7
MW: 192.2 D
From 60.00€ *
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S-Adenosylhomocysteine
S-Adenosylhomocysteine

Item number: Cay13603-50

S-Adenosyl-L-homocysteine (SAH) is an amino acid derivative and an intermediate, by-product, or modulator of several metabolic pathways, including the activated methyl cycle and cysteine biosynthesis. It is also a product of S-adenosyl-methionine (SAM)-dependent methylation of biological molecules, including DNA,...
Keywords: AdoHcy, SAH, S-(5'-deoxyadenosin-5'-yl)-L-homocysteine
Application: Metabolic studies
CAS 979-92-0
MW: 384.4 D
From 50.00€ *
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Valproic Acid (sodium salt)
Valproic Acid (sodium salt)

Item number: Cay13033-50

Valproic acid is an analog of the natural fatty acid valeric acid that inhibits class I histone deacetylases (HDACs) with an IC50 value of approximately 2 mM. It decreases the number of axon branches in sensory neurons isolated from newborn rat dorsal root ganglia, an effect that is reversed by...
Keywords: 2-Propylvaleric Acid, Valproate, VPA, 2-propyl-pentanoic acid, monosodium salt
Application: HDAC inhibitor
CAS 1069-66-5
MW: 166.2 D
From 50.00€ *
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Agomelatine
Agomelatine

Item number: Cay13203-50

Agomelatine is an agonist of melatonin (MT) receptors and a derivative of melatonin (Cay-14427). It binds to MT1 and MT2 receptors (Kis = 0.14 and 0.41 nM, respectively) and has an EC50 value of 0.1 nM in a [35S]GTPgammaS binding assay using CHO cells expressing MT2 receptors. Agomelatine is also an antagonist of...
Keywords: S20098, N-[2-(7-methoxy-1-naphthalenyl)ethyl]-acetamide
Application: Melatonin analog
CAS 138112-76-2
MW: 243.3 D
From 102.00€ *
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Lipoxin A4 methyl ester
Lipoxin A4 methyl ester

Item number: Cay10033-50

Lipoxin A4 (LXA4) methyl ester is a more lipid soluble, prodrug formulation of the transcellular metabolite LXA4. LXA4 is a trihydroxy fatty acid containing a conjugated tetraene, produced by the metabolism of 15-HETE or 15-HpETE with human leukocytes. LXA4 is equipotent to leukotriene B4 (LTB4) in inducing...
Keywords: 5(S),6(R),15(S)-TriHETE methyl ester, LXA4 methyl ester, 5S,6R,15S-trihydroxy-7E,9E,11Z,13E-eicosatetraenoic acid, methyl...
Application: Bioactive lipid assays
CAS 97643-35-1
MW: 366.5 D
From 368.00€ *
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Esomeprazole
Esomeprazole

Item number: Cay17303-50

Esomeprazole is an inhibitor of the gastric H+/K+-ATPase and the (S) enantiomer of omeprazole (Cay-14880). It reversibly inhibits the activity of the H+/K+-ATPase in an enzyme assay. Esomeprazole (30 mg/kg, s.c.) inhibits histamine-induced gastric acid secretion in rats. Formulations containing esomeprazole in...
Keywords: (-)-Omeprazole, (S)-Omeprazole, 6-methoxy-2-[(S)-[(4-methoxy-3,5-dimethyl-2-pyridinyl)methyl]sulfinyl]-1H-benzimidazole
Application: H+/K+-ATPase inhibitor
CAS 119141-88-7
MW: 345.4 D
From 43.00€ *
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