13 products were found matching "Cay13381"!

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CAY10606
CAY10606

Item number: Cay13381-5

5-Lipoxygenase (5-LO) initiates the synthesis of leukotrienes (LTs) from arachidonic acid, primarily in certain leukocyte populations. CAY10606 is a potent, reversible inhibitor of 5-LO, both in cell-free assays (IC50 = 86 nM) and in intact neutrophils (IC50 = 230 nM). It prevents the production of LTs in whole...
Keywords: 2-[(3-chlorophenyl)methyl]-5-hydroxy-1H-benz[g]indole-3-carboxylic acid, ethyl ester
Application: 5-LO inhibitor
CAS 1159576-98-3
MW: 379.8 D
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SU6656
SU6656

Item number: Cay13338-1

The Src family of proto-oncogenic kinases include nine mammalian non-receptor tyrosine kinases that are involved in intracellular signaling and are often relevant to carcinogenesis. SU6656 is a selective inhibitor of Src kinases, Including Src, Yes, Lyn, and Fyn (IC50 = 280, 20, 130, 170 nM, respectively). It weakly...
Keywords: 2,3-dihydro-N,N-dimethyl-2-oxo-3-[(4,5,6,7-tetrahydro-1H-indol-2-yl)methylene]-1H-indole-5-sulfonamide
Application: Src kinase inhibitor
CAS 330161-87-0
MW: 371.5 D
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2,4-Pyridinedicarboxylic Acid (hydrate)
2,4-Pyridinedicarboxylic Acid (hydrate)

Item number: Cay11138-1

2,4-Pyridinedicarboxylic Acid (2,4-PDCA) is a compound that structurally mimics 2-oxoglutarate (2-OG, also known as alpha-ketoglutarate) and chelates zinc, thus affecting a range of enzymes. As a 2-OG mimic, it blocks the activity of 2-OG oxygenases, which include certain lysine demethylases and a variety of...
Keywords: 2,4-Dicarboxylpyridine, 2,4-PDCA, 2,4-pyridinedicarboxylic acid, monohydrate
Application: 2-OG oxygenase inhibitor
CAS 207671-42-9
MW: 185.1 D
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K252a
K252a

Item number: Cay11338-1

K252a is a staurosporine analog isolated from Nocardiopsis sp. soil fungi that inhibits protein kinase (PK) C, PKA, Ca2+/calmodulin-dependent kinase type II, and phosphorylase kinase with IC50 values of 470, 140, 270, and 1.7 nM, respectively. Because it inhibits neurotrophin receptor tyrosine kinases, K252a at...
Keywords: SF 2370,...
Application: Kinase inhibitor
CAS 99533-80-9
MW: 467.5 D
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SR 9186
SR 9186

Item number: Cay13888-1

SR 9186 is an inhibitor of the cytochrome P450 (CYP) isoform CYP3A4 (IC50 = 0.011 µM). It is highly selective for CYP3A4 over CYP3A5 (IC50 = 33 µM). SR 9186 inhibits metabolism of midazolam to 1'-hydroxy midazolam, testosterone to 6beta-hydroxy testosterone, and vincristine to vincristine M1 in isolated human liver...
Keywords: N-(4'-cyano[1,1'-biphenyl]-4-yl)-N'-[4-(3H-imidazo[4,5-b]pyridin-7-yl)phenyl]-urea
Application: Selective CYP3A4 inhibitor
CAS 1361414-26-7
MW: 430.5 D
691.00€ *
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2-amino-4-phenyl Thiazole
2-amino-4-phenyl Thiazole

Item number: Cay13388-1

2-amino-4-phenyl Thiazole is a synthetic intermediate useful for pharmaceutical synthesis.Formal Name: 4-phenyl-2-thiazolamine. CAS Number: 2010-06-2. Synonyms: NSC 2528. Molecular Formula: C9H8N2S. Formula Weight: 176.2. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF:...
Keywords: NSC 2528, 4-phenyl-2-thiazolamine
Application: Synthetic intermediate, pharmaceutical synthesis
CAS 2010-06-2
MW: 176.2 D
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(1S,3S)-3-Hydroxycyclopentane acetic acid
(1S,3S)-3-Hydroxycyclopentane acetic acid

Item number: Cay11381-50

(1S,3S)-3-Hydroxycyclopentane acetic acid is a synthetic intermediate useful for pharmaceutical synthesis.Formal Name: 2-((1S,3S)-3-hydroxycyclopentyl)acetic acid. Molecular Formula: C7H12O3. Formula Weight: 144.2. Purity: >95%. Formulation: (Request formulation change), A neat oil. Solubility: DMF:, DMSO:,...
Keywords: 2-((1S,3S)-3-hydroxycyclopentyl)acetic acid
Application: Synthetic intermediate
MW: 144.2 D
114.00€ *
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DAz-2
DAz-2

Item number: Cay13382-1

DAz-2 is a cell-permeable chemical probe used to detect cysteine oxidation in proteins. Redox-sensitive cysteine residues in proteins may function as sensors of reactive oxygen species (ROS) and also serve as molecular switches, activating or deactivating proteins, following a change in oxidation state. Modification...
Keywords: Click Tag(TM) DAz-2, DCP-N3, 4-(3-azidopropyl)cyclohexane-1,3-dione
Application: Sulfenic acid probe
CAS 1176905-54-6
MW: 195.2 D
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2-methyl-4-phenyl Thiazole
2-methyl-4-phenyl Thiazole

Item number: Cay13386-1

2-methyl-4-phenyl Thiazole is a synthetic intermediate useful for pharmaceutical synthesis.Formal Name: 2-methyl-4-phenyl-thiazole. CAS Number: 1826-16-0. Molecular Formula: C10H9NS. Formula Weight: 175.3. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 25 mg/ml, DMSO:...
Keywords: 2-methyl-4-phenyl-thiazole
Application: Synthetic intermediate, Pharmaceutical synthesis
CAS 1826-16-0
MW: 175.3 D
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2-amino Pyridyl-5-thioamide
2-amino Pyridyl-5-thioamide

Item number: Cay13389-1

2-amino Pyridyl-5-thioamide is a synthetic intermediate useful for pharmaceutical synthesis.Formal Name: 6-amino-9-pyridinecarbothioamide. CAS Number: 53268-33-0. Molecular Formula: C6H7N3S. Formula Weight: 153.2. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 20...
Keywords: 6-amino-9-pyridinecarbothioamide
Application: Synthetic intermediate, Pharmaceutical synthesis
CAS 53268-33-0
MW: 153.2 D
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5-(2-Aminopyridyl)amide oxime
5-(2-Aminopyridyl)amide oxime

Item number: Cay13384-1

5-(2-Aminopyridyl)amide oxime is a synthetic intermediate useful for pharmaceutical synthesis.Formal Name: 6-amino-N-hydroxy-3-pyridinecarboximidamide. CAS Number: 468068-28-2. Molecular Formula: C6H8N4O. Formula Weight: 152.2. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility:...
Keywords: 6-amino-N-hydroxy-3-pyridinecarboximidamide
Application: Synthetic intermediate, Pharmaceutical synthesis
CAS 468068-28-2
MW: 152.2 D
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ethyl-2-amino-4-phenyl Thiophene-3-Carboxylate
ethyl-2-amino-4-phenyl Thiophene-3-Carboxylate

Item number: Cay13387-1

ethyl-2-amino-4-phenyl-Thiophene-3-carboxylate is a synthetic intermediate useful for pharmaceutical synthesis.Formal Name: ethyl ester-2-amino-4-phenyl-3-thiophenecarboxylic acid. CAS Number: 4815-36-5. Molecular Formula: C13H13NO2S. Formula Weight: 247.3. Purity: >98%. Formulation: (Request formulation change), A...
Keywords: ethyl ester-2-amino-4-phenyl-3-thiophenecarboxylic acid
Application: Synthetic intermediate, pharmaceutical synthesis
CAS 4815-36-5
MW: 247.3 D
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